BDBM50278337 CHEMBL470617::Naltrexone methiodide
SMILES C[N+]1(CC2CC2)CC[C@@]23[C@H]4Oc5c2c(C[C@@H]1[C@]3(O)CCC4=O)ccc5O
InChI Key InChIKey=JVLBPIPGETUEET-GAAHOAFPSA-O
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50278337
Affinity DataKi: 501nMAssay Description:Displacement of [3H]DPN from recombinant human delta opioid receptor expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]-DPN from recombinant human delta opioid receptor expressed in CHO-K1 cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.45E+3nMAssay Description:Displacement of [3H]-DADLE from human recombinant delta opioid receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.46E+3nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant delta opioid receptor assessed as reduction in SNC80 induced [3S]-GTPgammaS bindingMore data for this Ligand-Target Pair